Cmax (ng/mL) | Half-life (day-1) | F50 (ng/mL) | LC50D(TD) (ng/mL) | TD (days) | |
Macrocyclic lactones | |||||
Doramectin | 3.8:139.8 | 2.5:11.1 | 9.2 | 30.6 | 9 |
Eprinomectin | 3.4:503.0 | 1.0:5.7 | 1.0 | 7.6 | 9 |
Ivermectin | 2.7:316.0 | 0.4:7.8 | 4.1 | 7.3 | 9 |
Moxidectin | 2.6:420.0 | 1.4:23.1 | 478.4 | 1178.0 | 9 |
Isoxazolines | |||||
Afoxolaner | 621.9:1107.0 | 14.8:15.6 | 0* | 66.8 | 1 |
Fluralaner | 513.3:7109.0 | 11.0:18.6 | 0* | 21.2 | 1 |
Spinosyns | |||||
Spinosad | 1550.0 | 11.3 | 0* | 461.0 | 5 |
* remains to be measured for Anopheles.